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Research details

Difelikefalin — research data

Regulatory statusFDA-approved (Korsuva)
NCAA D1Not listed

Overview

About Difelikefalin

Mechanism of action

Selective peripherally restricted kappa opioid receptor agonist; reduces itch signaling

Safety profile

Dizziness, nausea, somnolence, falls · Approved for CKD pruritus; no classic opioid abuse potential; dizziness, diarrhea

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