Difelikefalin0 vendors competing
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Research details
Difelikefalin — research data
Regulatory statusFDA-approved (Korsuva)
NCAA D1Not listed
Overview
About Difelikefalin
Mechanism of action
Selective peripherally restricted kappa opioid receptor agonist; reduces itch signaling
Safety profile
Dizziness, nausea, somnolence, falls · Approved for CKD pruritus; no classic opioid abuse potential; dizziness, diarrhea
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